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EFIMOSFERMIN ALFA

UNII:Y114QW0F16
Type:INGREDIENT SUBSTANCE
Formula:
Preferred Substance Name:EFIMOSFERMIN ALFA
GSRS Full Record:

  • 2765640-39-7
  • BOS-580
  • EFIMOSFERMIN ALFA [USAN]
  • Efimosfermin Alfa
  • Efimosfermin alfa [WHO-DD]
  • Fc fragment of human immunoglobulin G1 (1-227) [Homo sapiens IGHG1*03 (hinge (1-10), CH2 L<sup>14</sup>>A, L<sup>15</sup> >A (11-120), CH3 (121-226), CHS (226-227))] fused via peptide linker <sup>228</sup>GS<sup>229</sup> to human fibroblast growth factor 21 (FGF-21) fragment 33-209 [Q<sup>55</sup> >C<sup>252</sup>, R<sup>105</sup> >K<sup>302</sup>, G<sup>148</sup> >C<sup>345</sup>, K<sup>150</sup> >R<sup>347</sup>, P<sup>158</sup> >S<sup>355</sup>, S<sup>195</sup> >A<sup>392</sup>, P<sup>199</sup> >G<sup>396</sup>, G<sup>202</sup> >A<sup>399</sup>]-variant (230-406 in the current sequence); dimer (6-6', 9-9')-bisdisulfide, produced in Chinese hamster ovary (CHO) cells, cell line CHO-DG44, glycoform alfa
  • Immunoglobulin G1 [14-alanine,15-alanine] (human γ1-chain C region C-terminal fragment) fusion protein with peptide linker (GS) fusion protein with 5-181-fibroblast growth factor 21 [27-cysteine,120-cysteine] (human), dimer
  • LLF-580
  • LLF580
  • efimosfermin alfa [INN]



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